Synthesis of substituted indazoles via [3+2] cycloaddition of benzyne and diazo compounds
CAS index name: 1H-indazole-3-carboxylic acid, ethyl ester
Organic SynthesesCycloaddition
A checked procedure from Organic Syntheses, the journal whose preparations are repeated in a second laboratory before publication. The full experimental, with amounts, hazards and characterisation data, is on orgsyn.org.
Reagents
| Compound | Role | Equiv | MW (g/mol) | ρ (g/mL) | Safety |
|---|---|---|---|---|---|
| Ethyl 3-indazolecarboxylate4498-68-4 · C10H10N2O2 | product | — | 190.20 | — | — |
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